211280
辣椒平
≥97% (HPLC), Capsaicin and resiniferatoxin antagonist, solid
别名:
辣椒平
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关于此项目
经验公式（希尔记法）:
C19H21ClN2O2S
化学文摘社编号:
分子量:
376.90
UNSPSC Code:
12352200
NACRES:
NA.77
MDL number:
产品名称
辣椒平, A competitive antagonist of Capsaicin and resiniferatoxin. Capsazepine (1 µM) blocks capsaicin (60 nM) stimulated firing of C-fibers.
Quality Level
assay
≥97% (HPLC)
form
solid
manufacturer/tradename
Calbiochem®
storage condition
OK to freeze
color
off-white
solubility
DMSO: soluble, methanol: soluble
shipped in
ambient
storage temp.
10-30°C
SMILES string
S=C(N2CCCc3c(cc(c(c3)O)O)C2)NCCc1ccc(cc1)Cl
InChI
1S/C19H21ClN2O2S/c20-16-5-3-13(4-6-16)7-8-21-19(25)22-9-1-2-14-10-17(23)18(24)11-15(14)12-22/h3-6,10-11,23-24H,1-2,7-9,12H2,(H,21,25)
InChI key
DRCMAZOSEIMCHM-UHFFFAOYSA-N
General description
感觉神经元兴奋剂辣椒素（目录编号211274）和树脂毒素（目录编号553975）的竞争性拮抗剂。辣椒素（1 µM）阻断辣椒素（60 nM）刺激的C纤维发射。
辣椒素（目录编号211274）和树脂毒素的竞争性拮抗剂。辣椒素（1 µM）阻断辣椒素（60 nM）刺激的C纤维发射。
Biochem/physiol Actions
主要靶标
辣椒素和树脂毒素的竞争性拮抗剂
辣椒素和树脂毒素的竞争性拮抗剂
产物不与ATP竞争。
可逆：否
细胞渗透性：否
Preparation Note
溶液中不稳定；仅在使用前进行复溶。
Other Notes
Fox, A.J., et al. 1995.Neuroscience 67, 741.
Ellis, J.L., and Undem, B.J.1994.J. Pharmacol.Exp.Ther.268, 85.
Walpole, C.S.J., et al. 1994.J. Med. Chem.37, 1942.
Szallasi, A., et al. 1993.J. Pharmacol.Exp.Therap.267, 728.
Ellis, J.L., and Undem, B.J.1994.J. Pharmacol.Exp.Ther.268, 85.
Walpole, C.S.J., et al. 1994.J. Med. Chem.37, 1942.
Szallasi, A., et al. 1993.J. Pharmacol.Exp.Therap.267, 728.
Legal Information
CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany
Disclaimer
毒性：标准处理（A）
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存储类别
11 - Combustible Solids
wgk
WGK 3
flash_point_f
Not applicable
flash_point_c
Not applicable
全球贸易项目编号
| 货号 | GTIN |
|---|---|
| 211280-10MG | 04055977219180 |