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M182

MDL-12,330A 盐酸盐

Name: MDL-12,330A 盐酸盐
Brand: SIGMA

≥98% (HPLC), Adenylyl cyclase inhibitor, powder

别名:

顺式-N-（2-苯基环戊基）-氮杂环十三碳-1-烯-2-胺盐酸盐

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关于此项目

经验公式（希尔记法）:

C₂₃H₃₆N₂ · HCl

化学文摘社编号:

40297-09-4

分子量:

377.01

UNSPSC Code:

41106305

PubChem Substance ID:

24896696

NACRES:

NA.77

MDL number:

MFCD00210204

Assay:

≥98% (HPLC)

Form:

powder

Quality level:

100

Storage condition:

desiccated

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属性

产品名称

MDL-12,330A 盐酸盐, ≥98% (HPLC), powder

Quality Level

100

assay

≥98% (HPLC)

form

powder

storage condition

desiccated

color

white to off-white

solubility

DMSO: >20 mg/mL

storage temp.

2-8°C

SMILES string

Cl[H].C1CCCCCN=C(CCCCC1)N[C@H]2CCC[C@H]2c3ccccc3

InChI

1S/C23H36N2.ClH/c1-2-4-6-11-18-23(24-19-12-7-5-3-1)25-22-17-13-16-21(22)20-14-9-8-10-15-20;/h8-10,14-15,21-22H,1-7,11-13,16-19H2,(H,24,25);1H/t21-,22-;/m0./s1

InChI key

CKOPQUCSDBVAQG-VROPFNGYSA-N

说明

Application

MDL-12,330A盐酸盐已用作腺苷酸环化酶抑制剂，抑制间充质干细胞(MSC)中的环磷腺苷信号传导。它也已用作腺苷酸环化酶抑制剂，检测其对悬尾实验(TST)小鼠自主活动的影响。

Biochem/physiol Actions

MDL-12,330A是一种环烷基内亚胺(lactamimide)，可用作电压门控钾离子通道阻断剂(KV)，有助于动作电位时程(APD)延长和胰岛素分泌。它也可阻断钙(Ca²⁺)内流通道。

腺苷酸环化酶抑制剂。

Features and Benefits

该化合物是受体分类及信号转导手册上腺苷酸环化酶页面上的特色化合物。想要浏览手册的其他页面，请单击此处。

这种化合物是环核苷酸研究的特色产品。点击此处发现更多特色环核苷酸产品。在sigma.com/discover-bsm可了解更多关于生物活性小分子的其他研究领域。

存储类别

11 - Combustible Solids

wgk

WGK 3

flash_point_f

Not applicable

flash_point_c

Not applicable

ppe

Eyeshields, Gloves, type N95 (US)

历史批次信息供参考:

分析证书(COA)

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全球贸易项目编号

货号	GTIN
M182-5MG	04061832898902
M182-25MG	04061832898896