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PZ0117

PF-573228

Name: PF-573228
Brand: SIGMA

≥95% (HPLC), FAK inhibitor, powder

别名:

6-[4-(3-(甲磺酰基-苄基-氨基)-5-三氟甲基-嘧啶-2-基氨基]-3,4-二氢-1H-喹啉-2-酮, PF-228

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关于此项目

经验公式（希尔记法）:

C₂₂H₂₀F₃N₅O₃S

化学文摘社编号:

869288-64-2

分子量:

491.49

UNSPSC Code:

12352200

PubChem Substance ID:

329823709

NACRES:

NA.77

MDL number:

MFCD11519967

Assay:

≥95% (HPLC)

Form:

powder

Quality level:

100

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属性

产品名称

PF-573228, ≥95% (HPLC)

Quality Level

100

assay

≥95% (HPLC)

form

powder

color

white to off-white

solubility

DMSO: ≥20 mg/mL

storage temp.

2-8°C

SMILES string

CS(=O)(=O)c1cccc(CNc2nc(Nc3ccc4NC(=O)CCc4c3)ncc2C(F)(F)F)c1

InChI

1S/C22H20F3N5O3S/c1-34(32,33)16-4-2-3-13(9-16)11-26-20-17(22(23,24)25)12-27-21(30-20)28-15-6-7-18-14(10-15)5-8-19(31)29-18/h2-4,6-7,9-10,12H,5,8,11H2,1H3,(H,29,31)(H2,26,27,28,30)

InChI key

HESLKTSGTIBHJU-UHFFFAOYSA-N

说明

Biochem/physiol Actions

PF-573228是一种粘着斑激酶（FAK）抑制剂；非受体酪氨酸激酶抑制剂。

Features and Benefits

该化合物是《受体分类及信号转导手册》上Fak页面上的特色化合物。想要浏览手册的其他页面，请单击此处。

这种化合物是激酶磷酸酶生物学研究的特色产品。点击此处发现更多特色激酶磷酸酶生物产品。在sigma.com/discover-bsm可了解更多关于生物活性小分子的其他研究领域。

pictograms

GHS07

signalword

Warning

hcodes

H302

pcodes

P264 - P270 - P301 + P312 - P501

Hazard Classifications

Acute Tox. 4 Oral

存储类别

11 - Combustible Solids

flash_point_f

Not applicable

flash_point_c

Not applicable

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